Megagrisevit Mono

Active Substance: Megagrisevit Mono

steroidinjectable

Description

What is Megagrisevit Mono?

Megagrisevit Mono is a brand name for the anabolic-androgenic steroid (AAS) clostebol acetate. Other names for this substance include:

  • 4-chlorotestosterone 17β-acetate (4-CLTA)

  • Macrobin

  • Steranabol

  • Alfa-Trofodermin

It is a synthetic derivative of testosterone and is typically administered via intramuscular injection. Clostebol acetate is designed to have a strong anabolic effect (promoting muscle growth) with a minimized androgenic effect (development of male sex characteristics).

Side Effects and Benefits

Benefits: In a medical context, clostebol acetate has been studied for its potential to:

  • Promote protein synthesis and nitrogen retention, which are key to muscle growth and repair.

  • Treat conditions where muscle wasting is a concern.

  • Increase red blood cell production.

However, the use of AAS for performance or image enhancement purposes is associated with significant and often severe side effects.

Side Effects: The side effects of anabolic steroids like clostebol acetate can be serious and wide-ranging. They can affect multiple body systems and may be long-lasting or irreversible.

  • Cardiovascular System: High blood pressure, blood clots, heart attacks, strokes, and damage to arteries. It can also negatively affect cholesterol levels by increasing "bad" LDL cholesterol and decreasing "good" HDL cholesterol.

  • Hormonal System (Men): Decreased sperm production, shrinking of the testicles (testicular atrophy), breast enlargement (gynecomastia), male-pattern baldness, and potential increase in testicular cancer risk.

  • Hormonal System (Women): Deepening of the voice, decreased breast size, excessive body hair growth (hirsutism), male-pattern baldness, and an enlarged clitoris. Some of these effects may be irreversible.

  • Liver: Oral forms of AAS can be particularly toxic to the liver, leading to liver tumors and blood-filled cysts (peliosis hepatis).

  • Psychiatric: Increased aggression ("roid rage"), mood swings, mania, and delusions.

  • Skin: Severe acne, oily skin, and potential abscesses at injection sites.

  • Musculoskeletal: In adolescents, it can cause bones to stop growing prematurely, resulting in stunted growth. It can also increase the risk of tendon injuries.

Pros and Cons

Pros:

  • Increased muscle mass and strength.

  • Improved athletic performance.

  • Potential therapeutic uses for specific medical conditions (under strict medical supervision).

Cons:

  • Severe and potentially irreversible side effects affecting the cardiovascular, hormonal, and liver systems.

  • Psychological and emotional side effects.

  • Risk of infection from non-sterile injection practices.

  • Illegality and ethical concerns in sports and other contexts.

Dosage and Frequency

Information regarding specific dosages for non-medical use is not publicly available or sanctioned. However, in a medical context, dosages would be carefully controlled by a physician. For its use in performance enhancement, clostebol acetate is often administered every two to three weeks, but this can vary depending on the specific use. It is crucial to understand that dosages used for non-medical purposes are often significantly higher than those prescribed therapeutically, leading to a much higher risk of adverse effects.

Half-Life and Detection Time

  • Half-Life: The half-life of a substance refers to the time it takes for half of the drug to be eliminated from the body. For clostebol acetate, the half-life is determined by how quickly the drug is absorbed from the injection site and then de-esterified in the body. The duration of the biological effects is determined by this absorption rate.

  • Detection Time: The detection time refers to how long a substance or its metabolites can be detected in a drug test, typically in urine or blood. For clostebol acetate, a single application can produce detectable metabolites in urine for more than 10 days. The precise detection window can vary based on the dosage, frequency of use, and the specific testing method used.

Sterogenic, Progestronic, and Prolactin Effects

  • Progestronic and Prolactin Effects: There is limited specific information available on the progestogenic and prolactin-related effects of clostebol acetate. However, some anabolic steroids can have progestogenic activity, which can lead to side effects like gynecomastia. Progestogenic compounds can also influence prolactin levels. It's important to note that the hormonal system is complex, and any steroid use can lead to a cascade of effects on various hormones, including those related to prolactin.

  • Sterogenic Effects: The term "sterogenic" is not a standard pharmacological term. Anabolic-androgenic steroids are a class of hormones based on the steroid nucleus. They exert their effects by interacting with androgen receptors and promoting protein synthesis.

Anabolic Androgenic Ratio

The anabolic-androgenic ratio is a way to compare the anabolic (muscle-building) effects of a steroid to its androgenic (masculinizing) effects. The ratio is relative to testosterone, which is often used as a baseline (1:1).

Clostebol acetate is specifically designed to have a more favorable anabolic-to-androgenic ratio than testosterone. This means it is intended to have a stronger anabolic effect relative to its androgenic effect, aiming to promote muscle growth while minimizing masculinizing side effects. However, a specific, universally accepted number for this ratio for clostebol acetate is not readily available in general public sources. Different studies or sources may report varying figures, but its primary purpose is to be "more anabolic and less androgenic" than testosterone.

Pharmacological Properties

Half Life

5 days

Active Dose

70%

Detection

3.57 weeks

Concentration

250 mg/ml

Anabolic/Androgenic Profile

Usage Effectiveness

Bulking
Cutting
Strength
Recomposition

Activity Profile

Estrogenic

None

Progestanic

None

Water Retention

None

Aromatization

No

Benefits

✓ Increased Muscle Mass ✓ Improved Strength Gains ✓ Enhanced Protein Synthesis ✓ Enhanced Athletic Performance ✓ Increased Red Blood Cell Production

Dosage Recommendations

Beginner

200-400 mg/week

Intermediate

400-600 mg/week

Advanced

600-800 mg/week

Side Effects

Common

⚠ Acne ⚠ Oily Skin ⚠ Hair Loss (Male Pattern Baldness) ⚠ Increased Body Hair Growth ⚠ Increased Blood Pressure ⚠ Mood Swings ⚠ Increased Aggression

Severe

⚠ Deepening of Voice (in females) ⚠ Virilization (in females) ⚠ Elevated Cholesterol (LDL) ⚠ Reduced HDL Cholesterol ⚠ Increased Risk of Blood Clots ⚠ Gynecomastia (Male Breast Enlargement) ⚠ Testicular Atrophy ⚠ Reduced Sperm Count ⚠ Liver Toxicity (Hepatotoxicity) ⚠ Abscess Formation

Safety Information

Liver Toxicity

None

Kidney Toxicity

Low

Cardiovascular Risk

Moderate

Disclaimer: This information is for educational purposes only. Always consult with a qualified healthcare professional before using any compounds.